SCHEMBL1044610

SCHEMBL1044610

NCCC1=CC(=O)NC1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15994560 0.98
Bromide SCHEMBL18044121 0.98
Acetic Acid SCHEMBL28734533 0.90
SCHEMBL1887392 0.87 HRH4 (0.31)
SCHEMBL1398019 0.85 GSK3A (0.32)
SCHEMBL31652590 0.85 MAOA (0.33)
Trifluoroacetic Acid SCHEMBL13722329 0.84 HRH4 (0.39)
SCHEMBL4174560 0.84 HRH1 (0.34)
SCHEMBL15228417 0.84 HRH1 (0.34)
Water SCHEMBL28158179 0.83 GSK3A (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 306 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220071917-A9 DRUG DELIVERY SYSTEMS AND METHODS COMPRISING POLYSIALIC ACID AND/OR OTHER POLYMERS UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2022-03-10 US claimed
CN-111514286-B Zika virus E protein conjugate vaccine and preparation method thereof 中国科学院过程工程研究所 2022-03-08 CN claimed
US-20210228494-A1 DRUG DELIVERY SYSTEMS AND METHODS COMPRISING POLYSIALIC ACID AND/OR OTHER POLYMERS UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2021-07-29 US claimed
EP-3703666-A1 DRUG DELIVERY SYSTEMS AND METHODS COMPRISING POLYSIALIC ACID AND/OR OTHER POLYMERS Universidade de Santiago de Compostela (ES) 2020-09-09 EP claimed
CN-109651224-A A kind of fluorescence protein crosslinking agent and preparation method thereof 苏州昊帆生物股份有限公司 2019-04-19 CN claimed
CN-104109201-B A kind of Exenatide18F labels and preparation method and application 江苏省原子医学研究所 2017-11-10 CN claimed
CN-104109201-A Exenatide &lt;18&gt;F marker, and preparation method and application thereof JIANGSU INST NUCLEAR MEDICINE 2014-10-22 CN claimed
US-20260102500-A1 PKC INHIBITORS FOR THE TREATMENT OF SEPTIC CHOLESTASIS WITH POLYMETHINE DYE TARGETING SMARTDYELIVERY GMBH (DE) 2026-04-16 US disclosed
EP-4720089-A1 COMPOSITIONS AND METHODS FOR IMAGING AND TREATING ENDOMETRIOSIS Endomet Biosciences, Inc. (US) 2026-04-08 EP disclosed
US-20260027227-A1 NOVEL THIOL REDUCTANT, METHOD AND USE THEREOF SUZHOU BIOREINNO BIOTECHNOLOGY LTD COMPANY (CN) 2026-01-29 US disclosed
US-20260022191-A1 METHOD OF PREPARING AN ANTIBODY WITH THIOL GROUP SITE-SPECIFIC MODIFICATIONS AND USE OF TCEP SUZHOU BIOREINNO BIOTECHNOLOGY LTD COMPANY (CN) 2026-01-22 US disclosed
US-20260015433-A1 METHOD OF PREPARING AN ANTIBODY WITH SITE-SPECIFIC MODIFICATIONS SUZHOU BIOREINNO BIOTECHNOLOGY LTD COMPANY (CN) 2026-01-15 US disclosed
US-20250354056-A1 POLYMER DOTS BIO RAD LABORATORIES INC (US) 2025-11-20 US disclosed
EP-1535952-A1 Method for preparing crosslinked polyelectrolyte multilayer films UNIVERSITE LOUIS PASTEUR (FR) 2005-06-01 EP disclosed
EP-1520176-A1 REAGENTS AND A METHOD FOR SATURATION LABELLING OF PROTEINS Amersham Biosciences UK Limited (GB) 2005-04-06 EP disclosed
WO-2004055117-A2 CARBOXAMIDE-SUBSTITUTED DYES FOR ANALYTICAL APPLICATIONS ATTO-TEC GMBH (DE) 2004-07-01 WO disclosed
WO-2004046170-A2 TUBULYSINS, METHOD FOR PRODUCING THE SAME AND TUBULYSIN PREPARATIONS GESELLSCHAFT FUER BIOTECHNOLOGISCHE FORSCHUNG MBH (GBF) (DE) 2004-06-03 WO disclosed
WO-2004005933-A1 REAGENTS AND A METHOD FOR SATURATION LABELLING OF PROTEINS AMERSHAM BIOSCIENCES UK LIMITED (GB) 2004-01-15 WO disclosed
US-6103236-A IN WHICH A COMPOUND HAVING AN AFFINITY FOR A TARGET CELL IS BOUND TO A TOXIN THROUGH A SPACER CONSISTING ESSENTIALLY OF POLYALKYLENE GLYCOL AND A DIPEPTIDE. KYOWA HAKKO KOGYO CO., LTD. (JP) 2000-08-15 US disclosed
EP-0867190-A1 NOVEL TOXIN COMPLEX KYOWA HAKKO KOGYO CO., LTD. (JP) 1998-09-30 EP disclosed