SCHEMBL10448362

SCHEMBL10448362

CC(C)(C)C(O[SiH3])[C@@H](O)C(OCc1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
KMT2A Q03164 1/20 0.36
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
CA1 P00915 2/20 0.34
MAPK1 P28482 2/20 0.33
MMP2 P08253 2/20 0.32
MMP3 P08254 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963799 0.77 ALDH1A1 (0.42) TRPA1KMT2AEDNRBEDNRACA1
SCHEMBL1059176 0.67 TSHR (0.40) KMT2ACA1TSHRHTTCA2
SCHEMBL1059178 0.67 TSHR (0.40) KMT2ACA1TSHRHTTCA2
SCHEMBL603883 0.67 CYP1A2 (0.45) MAPK1ALDH1A1LMNATSHR
SCHEMBL3855220 0.66 TSHR (0.46) CA1MAPK1ALDH1A1LMNATSHR
SCHEMBL9176021 0.66 MAPK1 (0.54) KMT2AMAPK1ALDH1A1TSHR
SCHEMBL5555540 0.65 TRPA1 (0.42) TRPA1KMT2ACA1MAPK1ALDH1A1
SCHEMBL1356758 0.64 TSHR (0.48) KMT2ACA1MAPK1ALDH1A1LMNA
SCHEMBL27905975 0.64 EDNRB (0.44) EDNRBEDNRAMAPK1ALDH1A1TSHR
SCHEMBL2959625 0.64 EDNRB (0.44) EDNRBEDNRAMAPK1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399743-A1 Phosphonomethylthio-alkoseypureine derivatives, intermediate products for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1990-11-28 EP disclosed