SCHEMBL10448705

SCHEMBL10448705

CN(NS(=O)(=O)Cc1ccccc1)S(=O)(=O)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
MMP1 P03956 1/20 0.52
MMP2 P08253 1/20 0.52
MMP9 P14780 1/20 0.52
MMP8 P22894 1/20 0.52
MMP13 P45452 1/20 0.52
HPGD P15428 4/20 0.47
HSD17B10 Q99714 2/20 0.47
USP2 O75604 1/20 0.47
HSP90AA1 P07900 1/20 0.47
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
HTT P42858 2/20 0.46
ALOX15 P16050 1/20 0.46
LMNA P02545 1/20 0.46
ADRB2 P07550 1/20 0.46
MAPT P10636 1/20 0.46
KDM4E B2RXH2 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10449151 0.83 KEAP1 (0.47) CA1CA2MMP1MMP2MMP9
SCHEMBL10448954 0.78 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1HTTLMNA
SCHEMBL3174757 0.77 HSP90AA1 (0.57) CA1CA2MMP1MMP2MMP9
SCHEMBL30988541 0.74 CA1 (0.55) CA1CA2MMP1MMP2MMP9
SCHEMBL7593278 0.73 PRSS1 (0.54) CA1CA2MMP1MMP2MMP9
SCHEMBL14951927 0.73 HSP90AA1 (0.53) CA1CA2MMP1MMP2MMP9
SCHEMBL13325 0.72 CA1 (0.63) CA1CA2MMP1MMP2MMP9
SCHEMBL6492175 0.72 CA1 (0.68) CA1CA2MMP1MMP2MMP9
SCHEMBL10900809 0.72 HSP90AA1 (0.52) CA1CA2MMP1MMP2MMP9
SCHEMBL11707925 0.72 HSP90AA1 (0.52) CA1CA2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4892887-A ANTITUMOR YALE UNIVERSITY (US) 1990-01-09 US disclosed
EP-0185387-B1 NOVEL, N,N'BIS(SULFONYL) HYDRAZINES HAVING ANTINEOPLASTIC ACTIVITY YALE UNIVERSITY (US) 1988-12-14 EP disclosed
US-4684747-A ANTITUMOR, ALKYLATING AGENTS YALE UNIVERSITY (US) 1987-08-04 US disclosed
EP-0185387-A1 Novel, N,N'bis(sulfonyl) hydrazines having antineoplastic activity YALE UNIVERSITY (US) 1986-06-25 EP disclosed