SCHEMBL10460596

SCHEMBL10460596

COc1cc(OCCCN2CCC(C(c3ccc(F)cc3)c3ccc(F)cc3)CC2)ccc1C(C)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.49
HTR2A P28223 3/20 0.49
MAOA P21397 2/20 0.49
KCNH2 Q12809 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 3/20 0.46
CYP2C9 P11712 2/20 0.46
HTR4 Q13639 2/20 0.46
USP2 O75604 1/20 0.46
HTR3E A5X5Y0 1/20 0.46
MLNR O43193 1/20 0.46
CACNA1F O60840 1/20 0.46
HTR3B O95264 1/20 0.46
HMGCR P04035 1/20 0.46
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46
DRD2 P14416 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
DRD1 P21728 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL10460538 0.97 MAOB (0.49) MAOBHTR2AMAOAMAPT
Oxalic Acid SCHEMBL10459285 0.89 HTR2A (0.49) HTR2ADRD3MAPT
SCHEMBL10556431 0.88 HTR2A (0.47) HTR2AUSP2HTR1ADRD2DRD1
SCHEMBL10560816 0.84 HRH2 (0.58) HTR2ACYP2D6HRH1
SCHEMBL10461368 0.83 PAX8 (0.59) MAOBMAOAKCNH2
SCHEMBL7320146 0.83 ABCB11 (0.61) HTR2AKCNH2HTR1AADRA2ADRD2
SCHEMBL10558384 0.83 HTR2A (0.53) HTR2AUSP2HTR1ADRD2DRD1
Hydrochloric Acid SCHEMBL10459192 0.83 PAX8 (0.58) MAOBMAOAKCNH2
SCHEMBL10461614 0.82 HTR2A (0.47) MAOBHTR2AUSP2HTR1ADRD2
SCHEMBL10460536 0.81 HTR2A (0.58) HTR2AUSP2HTR1ADRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US claimed