SCHEMBL10464937

SCHEMBL10464937

CCNS(=O)(=O)c1nc2ccccc2n1CC(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
CTSD P07339 5/20 0.54
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ALDH1A1 P00352 2/20 0.50
NPSR1 Q6W5P4 3/20 0.49
POLB P06746 1/20 0.49
RAB9A P51151 2/20 0.47
MAPK1 P28482 1/20 0.47
CXCR3 P49682 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MAPT P10636 1/20 0.47
GUSB P08236 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10465055 0.86 POLB (0.52) HTTCYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL10466119 0.84 CTSD (0.47) HTTCTSDALDH1A1POLBRAB9A
SCHEMBL10466200 0.82 POLB (0.67) HTTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6325602 0.75 SMN1; SMN2 (0.70) HTTCTSDCYP1A2CYP2D6CYP2C9
SCHEMBL8565487 0.69 SMN1; SMN2 (1.00) SMN1; SMN2ALDH1A1NPSR1POLBRAB9A
SCHEMBL8563635 0.68 SMN1; SMN2 (0.80) CYP1A2CYP2D6CYP2C9CYP2C19SMN1; SMN2
Bromide SCHEMBL8864660 0.68 SMN1; SMN2 (0.97) SMN1; SMN2ALDH1A1NPSR1POLBRAB9A
SCHEMBL9568271 0.68 SMN1; SMN2 (0.86) SMN1; SMN2ALDH1A1NPSR1POLB
Hydrochloric Acid SCHEMBL8864540 0.68 SMN1; SMN2 (0.78) CYP1A2CYP2D6CYP2C9CYP2C19SMN1; SMN2
Bromide SCHEMBL8864504 0.67 SMN1; SMN2 (0.84) SMN1; SMN2ALDH1A1NPSR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0246126-A1 Benzimidazoles and imidazopyridine sulfone amides, process for their preparation and their use as medicaments LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1987-11-19 EP claimed
US-4943570-A GASTROINTESTINAL DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1990-07-24 US disclosed
US-4933338-A ANTIULCER AGENTS, ANTISECRETORY AGENTS, TREATMENT OF GASTROINTESTINAL DISORDERS; CHEMICAL INTERMEDIATES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1990-06-12 US disclosed
EP-0246126-A1 Benzimidazoles and imidazopyridine sulfone amides, process for their preparation and their use as medicaments LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1987-11-19 EP disclosed