SCHEMBL10474167

SCHEMBL10474167

Cn1c(-c2c(F)cccc2F)nn(-c2ccccc2Br)c1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.43
BTK Q06187 1/20 0.43
OPRM1 P35372 1/20 0.41
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
MGLL Q99685 2/20 0.37
KCNN4 O15554 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HCAR1 Q9BXC0 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
WNT3A P56704 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10473916 0.91 JAK2 (0.40) JAK2BTKOPRM1ALDH1A1SMN1; SMN2
SCHEMBL10474202 0.82 HSD11B1 (0.43) KCNN4ALDH1A1HCAR1L3MBTL1
SCHEMBL7652883 0.80 OPRM1 (0.41) OPRM1GSK3AGSK3BMGLLALDH1A1
SCHEMBL10475264 0.80 HCAR1 (0.39) JAK2BTKALDH1A1SMN1; SMN2HCAR1
SCHEMBL10474070 0.76 CDK4 (0.38) ALDH1A1SMN1; SMN2
SCHEMBL7658070 0.74 NPC1 (0.44) MGLLALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL10475265 0.72 MAPT (0.38) ALDH1A1L3MBTL1
SCHEMBL10475053 0.71 OPRM1 (0.36) JAK2BTKOPRM1MGLLKCNN4
SCHEMBL10475378 0.71 GAA (0.46) ALDH1A1L3MBTL1
SCHEMBL30582372 0.69 DHODH (0.40) OPRM1GSK3AGSK3BMGLLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4943583-A PESTICIDES HOFFMANN-LA ROCHE INC. (US) 1990-07-24 US disclosed
EP-0270061-A2 Five-membered heterocycles with three heteroatoms, their preparation and their use as pesticides CIBA-GEIGY AG (CH) 1988-06-08 EP disclosed