SCHEMBL10474202

SCHEMBL10474202

Cn1c(-c2c(F)cccc2F)nn(-c2ccccc2C(F)(F)F)c1=O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.43
SCN9A Q15858 1/20 0.41
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.38
KCNN4 O15554 1/20 0.38
POLB P06746 1/20 0.38
MDM2 Q00987 1/20 0.38
DHODH Q02127 5/20 0.37
HCAR1 Q9BXC0 2/20 0.37
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10473909 0.85 HSD11B1 (0.43) HSD11B1SCN9AALDH1A1L3MBTL1KCNN4
SCHEMBL10475020 0.82 ALDH1A1 (0.38) HSD11B1SCN9AALDH1A1L3MBTL1GAA
SCHEMBL10474167 0.82 JAK2 (0.43) ALDH1A1L3MBTL1KCNN4HCAR1
SCHEMBL10475264 0.78 HCAR1 (0.39) SCN9AALDH1A1GAAATMDHODH
SCHEMBL10474147 0.77 HSD11B1 (0.61) HSD11B1GAAATMMAPK14
SCHEMBL10474070 0.74 CDK4 (0.38) ALDH1A1GAAATMDHODHMAPK14
SCHEMBL10473916 0.74 JAK2 (0.40) HSD11B1ALDH1A1L3MBTL1GAAATM
SCHEMBL10595769 0.74 ALDH1A1 (0.40) HSD11B1SCN9AALDH1A1L3MBTL1GAA
SCHEMBL10475055 0.73 MGLL (0.41) SCN9AALDH1A1L3MBTL1KCNN4POLB
SCHEMBL10475137 0.73 MAPT (0.41) SCN9AALDH1A1L3MBTL1GAAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4943583-A PESTICIDES HOFFMANN-LA ROCHE INC. (US) 1990-07-24 US disclosed
EP-0270061-A2 Five-membered heterocycles with three heteroatoms, their preparation and their use as pesticides CIBA-GEIGY AG (CH) 1988-06-08 EP disclosed