SCHEMBL10474175

SCHEMBL10474175

O=Cc1c(Cl)nc2ccccc2c1-c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.46
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
PRKAA2 P54646 1/20 0.43
GRM2 Q14416 1/20 0.43
ADORA2A P29274 1/20 0.42
KDM4E B2RXH2 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NR1I2 O75469 1/20 0.41
NR4A2 P43354 1/20 0.41
PDE4D Q08499 1/20 0.41
ALOX5 P09917 1/20 0.40
ERN1 O75460 1/20 0.39
HMGCR P04035 1/20 0.39
HPGD P15428 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474212 0.80 KDM4E (0.46) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL8321756 0.80 GCGR (0.46) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL29419163 0.79 RXRA (0.67) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL244423 0.79 RXRA (0.67) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL28261499 0.78 RXRA (0.44) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL27560748 0.77 RXRA (0.62) RXRATNKSTNKS2PARP2PRKAA2
SCHEMBL11359732 0.77 ADORA2A (0.44) TNKSTNKS2PARP2GRM2ADORA2A
SCHEMBL4860650 0.75 MAOA (0.55) KDM4ERXFP1PDE4DERN1NPSR1
SCHEMBL10475261 0.74 PRKAA2 (0.66) TNKSTNKS2PARP2PRKAA2GRM2
SCHEMBL23780919 0.72 ERN1 (0.45) KDM4ERXFP1PDE4DERN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4923861-A 6-(2-(2-(Substituted amino)-3-quinolinyl) ethenyl and ethyl) tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed