SCHEMBL10487486

SCHEMBL10487486

BrC[C@@H](Cc1ccccc1)Oc1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.43
PPARA Q07869 15/20 0.43
SLC6A4 P31645 1/20 0.41
LDHA P00338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818873 0.85 PPARG (0.46) PPARGPPARALDHA
SCHEMBL11292923 0.77 PPARG (0.50) PPARGPPARA
SCHEMBL10487454 0.76 RAB9A (0.51) PPARGPPARA
SCHEMBL27617197 0.76 SIGMAR1 (0.46) SLC6A4
SCHEMBL106764 0.75 EPHX1 (0.44) SLC6A4
SCHEMBL11757844 0.75 PPARG (0.42) PPARGPPARA
SCHEMBL11659888 0.75 TSHR (0.39) PPARGPPARASLC6A4
SCHEMBL9818821 0.73 PPARG (0.76) PPARGPPARA
SCHEMBL7001784 0.73 MAOA (0.53) PPARGPPARA
SCHEMBL10487481 0.72 PPARG (0.61) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4853410-A Hydroxyacetic acid derivatives for the treatment of diabetic complications PFIZER INC. (US) 1989-08-01 US disclosed
WO-1987004344-A1 HYDROXYACETIC ACID DERIVATIVES FOR THE TREATMENT OF DIABETIC COMPLICATIONS PFIZER INC. (US) 1987-07-30 WO disclosed
EP-0230379-A2 Chroman- and thiochroman-4-acetic acids useful in the treatment of diabetic complications PFIZER INC. (US) 1987-07-29 EP disclosed