SCHEMBL10500751

SCHEMBL10500751

Cn1c(=O)c2c(ncn2CCNCc2ccccc2)n(C)c1=O

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.71
ADORA2B P29275 7/20 0.69
SMN1; SMN2 Q16637 2/20 0.69
RXFP1 Q9HBX9 1/20 0.69
TSHR P16473 2/20 0.68
CNOT7 Q9UIV1 1/20 0.60
LMNA P02545 2/20 0.56
MAPT P10636 1/20 0.56
GLA P06280 1/20 0.55
HTT P42858 1/20 0.55
UBE2N P61088 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
MAPK1 P28482 1/20 0.54
POLB P06746 1/20 0.53
HIF1A Q16665 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10501627 0.94 TSHR (0.74) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
SCHEMBL10178175 0.89 LMNA (0.56) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
Pimefylline SCHEMBL363878 0.88 LMNA (0.70) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
Pimefylline SCHEMBL29974579 0.88 LMNA (0.70) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
SCHEMBL4480581 0.84 ALDH1A1 (0.56) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
Benzene SCHEMBL27777114 0.84 ADORA2B (0.64) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
Toluene SCHEMBL28070325 0.83 ALDH1A1 (0.61) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
SCHEMBL17786242 0.83 ALDH1A1 (1.00) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
Pimefylline SCHEMBL9252493 0.82 LMNA (0.65) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR
SCHEMBL1944405 0.82 ADORA2B (1.00) ALDH1A1ADORA2BSMN1; SMN2RXFP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167008-B1 1,4:3,6-DIANHYDRO-HEXITE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS Heinrich Mack Nachf. (DE) 1989-09-06 EP disclosed
US-4769379-A Dianhydrohexite derivatives, and their use as pharmaceuticals HEINRICH MACK NACHF. (DE) 1988-09-06 US disclosed
EP-0167008-A2 1,4:3,6-Dianhydro-hexite derivatives, process for their preparation and their use as medicaments Heinrich Mack Nachf. (DE) 1986-01-08 EP disclosed
US-4150227-A Process for the production of basic substituted alkyl theophylline DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1979-04-17 US disclosed