SCHEMBL1051771

SCHEMBL1051771

COCCCc1c[nH]c2ccc(C(C)C(CC(C(O)CNC(C)C)N(C(=O)O)C(C)(C)C)C(C)C)cc12

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.33
HTR1D P28221 5/20 0.33
HTR1B P28222 4/20 0.33
MTNR1A P48039 4/20 0.32
MTNR1B P49286 3/20 0.32
KMT2A Q03164 2/20 0.32
TRPV1 Q8NER1 2/20 0.32
PTGS2 P35354 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SPR P35270 1/20 0.31
POLB P06746 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1051390 0.91 ACHE (0.34) ACHEHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL1050938 0.90 HTR1D (0.37) ACHEHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL5050472 0.84 HTR1D (0.35) HTR1DHTR1BMTNR1AMTNR1BKMT2A
SCHEMBL1051032 0.84 HTR1D (0.36) ACHEHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL1049206 0.83 HTR1D (0.36) ACHEHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL1049543 0.82 HTR1D (0.39) HTR1DHTR1BMTNR1AMTNR1BTRPV1
Hydrochloric Acid SCHEMBL1049681 0.82 HTR1D (0.39) HTR1DHTR1BMTNR1AMTNR1BKMT2A
SCHEMBL1049891 0.77 MTNR1A (0.35) MTNR1AMTNR1BKMT2ATRPV1PTGS2
Hydrochloric Acid SCHEMBL1050543 0.76 TRPV1 (0.36) HTR1DMTNR1AMTNR1BKMT2ATRPV1
SCHEMBL4533872 0.76 HTR1D (0.31) HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868036-B2 Organic compounds NOVARTIS AG (CH) 2011-01-11 US disclosed