SCHEMBL10534331

SCHEMBL10534331

Clc1ccc2c(c1)CCC(c1ccccc1)S2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
GRIN2B Q13224 1/20 0.38
TRPM4 Q8TD43 2/20 0.37
TRPM5 Q9NZQ8 2/20 0.37
ALOX12 P18054 1/20 0.37
TP53 P04637 1/20 0.34
MDM2 Q00987 1/20 0.34
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GSK3B P49841 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ATM Q13315 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
FADS1 O60427 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CYP2A6 P11509 1/20 0.33
HTT P42858 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10534373 0.92 BCHE (0.35) KDM1AMAOAMAOBGRIN2BTP53
SCHEMBL9565775 0.83 TRPM5 (0.41) TRPM4TRPM5ALOX12TP53HPGD
SCHEMBL11099067 0.83 ESR1 (0.41) KDM1AMAOAMAOBTP53MDM2
SCHEMBL10534797 0.80 PRCP (0.41) GSK3BSMN1; SMN2HTR2AHTR2CSIGMAR1
SCHEMBL44650 0.79 SIGMAR1 (0.44) KDM1AMAOAMAOBGRIN2BGSK3B
SCHEMBL24899246 0.70 KDM1A (0.49) KDM1AMAOAMAOBTRPM4TRPM5
SCHEMBL22072985 0.70 KDM1A (0.49) KDM1AMAOAMAOBTRPM4TRPM5
SCHEMBL27909263 0.70 KDM1A (0.49) KDM1AMAOAMAOBTRPM4TRPM5
SCHEMBL10534782 0.70 HPGD (0.49) TP53HPGDL3MBTL1GSK3BSMN1; SMN2
SCHEMBL6414384 0.67 TSHR (0.36) KDM1AMAOAMAOBSMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4801593-A VIRICIDE FOR RHINITIS VIRUS CONTAINING 2-PHENYLTETRALIN DERIVATIVE BURROUGHS WELLCOME CO. (US) 1989-01-31 US disclosed
EP-0025598-B1 THE USE OF 2-PHENYLTETRALIN DERIVATIVES, OR HETEROCYCLIC ANALOGUES, IN MEDICINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1984-08-01 EP disclosed
EP-0025598-A1 The use of 2-phenyltetralin derivatives, or heterocyclic analogues, in medicine and pharmaceutical compositions containing them THE WELLCOME FOUNDATION LIMITED (GB) 1981-03-25 EP disclosed