SCHEMBL10551908

SCHEMBL10551908

COc1cc([S+](C)[O-])ccc1-c1nc2cc3c(cc2[nH]1)[nH]c(=O)n3C

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 8/20 0.39
LMNA P02545 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
TP53 P04637 2/20 0.37
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
PDE5A O76074 1/20 0.37
PDE2A O00408 1/20 0.35
BRD4 O60885 2/20 0.34
CCR4 P51679 1/20 0.34
BRPF1 P55201 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705442 0.88 KDM4E (0.41) AMY1AKDM4ECYP1A2CYP3A4PDE3B
SCHEMBL10552590 0.85 TP53 (0.38) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL9703649 0.83 AMY1A (0.43) AMY1ATP53PDE3BPDE3APDE5A
SCHEMBL10552928 0.83 CDK4 (0.45) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL10552771 0.82 KDM4E (0.40) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL10551871 0.82 AMY1A (0.40) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL9678840 0.79 KDM4E (0.43) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL10552087 0.79 AMY1A (0.38) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL10554215 0.78 AMY1A (0.38) AMY1ALMNAKDM4ECYP1A2CYP3A4
SCHEMBL9702924 0.78 AMY1A (0.41) AMY1ALMNAKDM4ECYP1A2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831032-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE, ISOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1989-05-16 US disclosed