SCHEMBL10554666

SCHEMBL10554666

C=CC(=O)N(C)C(=O)C=Cc1ccc(C)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 4/20 0.54
MAPT P10636 5/20 0.50
RAB9A P51151 2/20 0.49
KMT2A Q03164 1/20 0.49
FOS P01100 1/20 0.47
JUN P05412 1/20 0.47
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
POLB P06746 1/20 0.45
SLC5A1 P13866 1/20 0.43
SLC5A2 P31639 1/20 0.43
CYP1B1 Q16678 1/20 0.42
HSD17B3 P37058 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877335 0.79 TRPM8 (0.60) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL9302644 0.77 TRPM8 (0.58) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL9302651 0.77 TRPM8 (0.58) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL25199560 0.77 FOS (0.65) TRPM8MAPTRAB9AKMT2AFOS
Acrylic Acid SCHEMBL6862453 0.75 KDM4E (0.59) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL10777127 0.75 TRPM8 (0.55) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL26186292 0.74 SMN1; SMN2 (0.57) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL28501196 0.72 NPC1 (0.72) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL10271039 0.72 TRPM8 (0.74) TRPM8MAPTRAB9AKMT2AFOS
SCHEMBL11217696 0.72 HSD17B3 (0.55) TRPM8MAPTRAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4883877-A CALCIUM METABOLISM REGULATORS, INHIBIT BONE RESORPTION, ANTIARTHRITIC CIBA-GEIGY CORPORATION (US) 1989-11-28 US disclosed
EP-0317506-A2 Azabicycloheptanes and method for their preparation CIBA-GEIGY AG (CH) 1989-05-24 EP disclosed