SCHEMBL10567017

SCHEMBL10567017

CC(=O)C1C(=O)Nc2cc3[nH]c(-c4ncc[nH]4)nc3cc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.34
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GAA P10253 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
ATM Q13315 1/20 0.31
ERAP1 Q9NZ08 1/20 0.31
PARP1 P09874 1/20 0.31
TBK1 Q9UHD2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10733805 0.81 PGR (0.35) IDO1KDM4EALDH1A1HPGDNPC1
SCHEMBL9830544 0.81 PDE4A (0.51) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL9832544 0.78 CHRNB2 (0.42) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL9833850 0.78 ALDH1A1 (0.53) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL10373859 0.76 CHEK2 (0.49) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL10567045 0.71 TLK2 (0.30)
SCHEMBL10767730 0.70 CHRNB2 (0.37) ALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL9832273 0.70 PDE4A (0.48) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL10372601 0.69 PDE2A (0.36) KDM4ETP53PDE3BPDE3A
SCHEMBL10373839 0.69 CYP17A1 (0.40) KDM4EALDH1A1HPGDRAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed