SCHEMBL10567136

SCHEMBL10567136

CC1(C)C(=O)Nc2cc3c(cc21)NC(Cc1cccs1)N3

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.45
MAPT P10636 1/20 0.43
PDK2 Q15119 1/20 0.38
PDK4 Q16654 1/20 0.38
ATAD2 Q6PL18 1/20 0.37
PGR P06401 6/20 0.35
PDE4A P27815 6/20 0.34
PDE4B Q07343 6/20 0.34
PDE4C Q08493 6/20 0.34
PDE4D Q08499 6/20 0.34
PDE3B Q13370 6/20 0.34
PDE3A Q14432 6/20 0.34
HDAC2 Q92769 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833683 0.78 PDE3B (0.46) PDK2PDK4ATAD2PGRPDE4A
SCHEMBL10566335 0.78 ALDH1A1 (0.49) HSD17B10MAPTPDK2PDK4ATAD2
Water SCHEMBL10471047 0.77 PDE3B (0.45) PDK2PDK4ATAD2PGRPDE4A
SCHEMBL10701189 0.77 HSD17B10 (0.41) HSD17B10MAPTHDAC2HDAC8HDAC6
SCHEMBL9835356 0.75 ATAD2 (0.46) PDK2PDK4ATAD2PGRPDE4A
SCHEMBL10695728 0.74 MAPT (0.39) HSD17B10MAPTHDAC2HDAC8HDAC6
SCHEMBL9833110 0.74 GSK3B (0.46) HSD17B10PDK2PDK4ATAD2PGR
SCHEMBL9834972 0.73 ATAD2 (0.50) PDK2PDK4ATAD2PGRPDE4A
SCHEMBL9835634 0.73 ATAD2 (0.44) PDK2PDK4ATAD2PGRPDE4A
SCHEMBL10668135 0.72 ATAD2 (0.43) PDK2PDK4ATAD2PGRPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed