SCHEMBL9833110

SCHEMBL9833110

CC1(C)C(=O)Nc2cc3c(cc21)NC(Cc1cccnc1)N3

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.46
PDE4A P27815 3/20 0.38
PDE4B Q07343 3/20 0.38
PDE4C Q08493 3/20 0.38
PDE4D Q08499 3/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
PDK2 Q15119 1/20 0.37
PDK4 Q16654 1/20 0.37
MMP1 P03956 2/20 0.37
MAOB P27338 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ATAD2 Q6PL18 1/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HRH4 Q9H3N8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10472432 0.90 GSK3B (0.39) GSK3BPDE4APDE4BPDE4CPDE4D
SCHEMBL9833683 0.85 PDE3B (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
Water SCHEMBL10471047 0.84 PDE3B (0.45) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL6455942 0.77 DDB1 (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835356 0.74 ATAD2 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10567136 0.74 HSD17B10 (0.45) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834421 0.74 ALDH1A1 (0.41) TSHRKDM4EALDH1A1PGR
SCHEMBL9832061 0.72 PDE3B (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835634 0.72 ATAD2 (0.44) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833102 0.71 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed