SCHEMBL10568563

SCHEMBL10568563

N#CCc1ccccc1Cc1ccccc1O

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 1/20 0.64
KEAP1 Q14145 1/20 0.47
TSHR P16473 2/20 0.42
CYP2D6 P10635 1/20 0.42
HIF1A Q16665 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
AKR1B1 P15121 1/20 0.41
CA12 O43570 5/20 0.39
CA2 P00918 5/20 0.39
IDO1 P14902 2/20 0.39
CA9 Q16790 4/20 0.38
MPO P05164 1/20 0.38
HTR1A P08908 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL891289 0.87 HSPA5 (0.54) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL8763318 0.87 ALDH1A1 (0.50) HSPA5TSHRALDH1A1HPGDKDM4E
SCHEMBL7809667 0.82 HSPA5 (0.94) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL5852726 0.82 HSPA5 (0.94) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL4003141 0.81 KEAP1 (0.63) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL1945874 0.80 ALDH1A1 (0.56) TSHRALDH1A1HPGDKDM4E
SCHEMBL29809738 0.80 ALDH1A1 (0.56) TSHRALDH1A1HPGDKDM4E
SCHEMBL49745 0.80 HSPA5 (1.00) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL29357407 0.80 HSPA5 (1.00) HSPA5KEAP1TSHRCYP2D6HIF1A
SCHEMBL29839938 0.78 HSPA5 (0.94) HSPA5KEAP1TSHRCYP2D6HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4874763-A ANTIARRHYTHMIA AGENTS ROEHM GMBH CHEMISCHE FABRIK (DE) 1989-10-17 US disclosed
EP-0318795-A2 Pharmaceutically active pteridin derivatives Röhm GmbH (DE) 1989-06-07 EP disclosed