SCHEMBL1060208

SCHEMBL1060208

CC(C)N(C(C)C)P(OCC(Cl)(Cl)Cl)N(C(C)C)C(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15682915 0.79
SCHEMBL22801231 0.74
SCHEMBL14064163 0.72
SCHEMBL15557296 0.71
SCHEMBL7572703 0.70 LMNA (0.30)
SCHEMBL10138045 0.65
SCHEMBL24945919 0.65
SCHEMBL6439415 0.65
SCHEMBL20343302 0.65
SCHEMBL13801800 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112979695-B Method for preparing 1, 2-di-fatty acyl-sn-glycerol-3-phosphatidylserine 苏州昊帆生物股份有限公司 2022-04-12 CN claimed
US-10414790-B2 Exocyclic nitrogen atom protected nucleoside and method for producing and using the same THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2019-09-17 US claimed
US-20150225442-A1 EXOCYLIC NITROGEN ATOM PROTECTED NUCLEOSIDE AND METHOD FOR PRODUCING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2015-08-13 US claimed
WO-2014022839-A1 EXOCYLIC NITROGEN ATOM PROTECTED NUCLOSIDE AND METHOD FOR PRODUCING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2014-02-06 WO claimed
WO-2025063239-A1 SIRNA CAPABLE OF SUPPRESSING EXPRESSION OF α-SYNUCLEIN 第一三共株式会社 2025-03-27 WO disclosed
WO-2025063238-A1 SIRNA FOR SUPPRESSING EXPRESSION OF PHOSPHOLAMBAN 第一三共株式会社 2025-03-27 WO disclosed
CN-112979695-B Method for preparing 1, 2-di-fatty acyl-sn-glycerol-3-phosphatidylserine 苏州昊帆生物股份有限公司 2022-04-12 CN disclosed
CN-112979695-B Method for preparing 1, 2-di-fatty acyl-sn-glycerol-3-phosphatidylserine 苏州昊帆生物股份有限公司 2022-04-12 CN disclosed
US-10414790-B2 Exocyclic nitrogen atom protected nucleoside and method for producing and using the same THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2019-09-17 US disclosed
US-20150225442-A1 EXOCYLIC NITROGEN ATOM PROTECTED NUCLEOSIDE AND METHOD FOR PRODUCING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2015-08-13 US disclosed
US-8957201-B2 Oligonucleotide analogues and methods utilizing the same DAIICHI SANKYO COMPANY, LIMITED (JP) 2015-02-17 US disclosed
WO-2014022839-A1 EXOCYLIC NITROGEN ATOM PROTECTED NUCLOSIDE AND METHOD FOR PRODUCING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2014-02-06 WO disclosed
US-20090149404-A1 Oligonucleotide analogues and methods utilizing the same DAIICHI SANKYO COMPANY, LIMITED (JP) 2009-06-11 US disclosed
US-7335765-B2 Nucleoside and oligonucleotide analogues DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-02-26 US disclosed
US-7314923-B2 Nucleoside and oligonucleotide analogues DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-01 US disclosed
US-20050261235-A1 2' ,5' -Oligoadenylate analogs SANKYO COMPANY, LIMITED (JP) 2005-11-24 US disclosed
EP-1568704-A1 NOVEL 2' ,5' -OLIGOADENYLIC ACID ANALOGUES Sankyo Company, Limited (JP) 2005-08-31 EP disclosed
US-20030207841-A1 Novel nucleoside and oligonucleotide analogues SANKYO COMPANY LIMITED (JP) 2003-11-06 US disclosed
US-20020147332-A1 Novel nucleoside and oligonucleotide analogues SANKYO COMPANY, LIMITED (JP) 2002-10-10 US disclosed
EP-1152009-A1 NOVEL NUCLEOSIDES AND OLIGONUCLEOTIDE ANALOGUES Sankyo Company, Limited (JP) 2001-11-07 EP disclosed