SCHEMBL10622656

SCHEMBL10622656

CSCC[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.62
CTSK P43235 6/20 0.62
REN P00797 1/20 0.53
CA2 P00918 1/20 0.51
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
ACE P12821 1/20 0.48
CCKBR P32239 1/20 0.48
LTA4H P09960 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10622674 1.00 CTSS (0.62) CTSSCTSKRENCA2CTSL
SCHEMBL7815002 0.91 REN (0.61) CTSSCTSKRENCTSLCTSB
SCHEMBL11443643 0.90 ITGB3 (0.52) CTSSCTSKRENCA2CTSL
SCHEMBL11123415 0.89 CTSS (0.62) CTSSCTSKRENCA2CTSL
SCHEMBL28630396 0.89 CTSS (0.72) CTSSCTSKRENCTSLCTSB
SCHEMBL10144086 0.88 CTSS (0.55) CTSSCTSKRENCA2CCKBR
SCHEMBL11605396 0.88 CTSS (0.56) CTSSCTSKRENCA2CTSL
SCHEMBL11606668 0.88 CTSS (0.56) CTSSCTSKRENCA2CTSL
SCHEMBL11333258 0.87 CTSS (0.59) CTSSCTSKRENCA2CTSL
SCHEMBL11105884 0.87 ACE (0.61) CTSSCTSKRENCA2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4757153-A Substituted phenyl group containing pharmaceuticals G. D. SEARLE & CO. (US) 1988-07-12 US disclosed
EP-0212550-A2 Substituted dipeptide amides G.D. Searle & Co. (US) 1987-03-04 EP disclosed