SCHEMBL10642802

SCHEMBL10642802

OC(O)C1CN(Cc2ccccc2)C1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FUCA1 P04066 2/20 0.65
SIGMAR1 Q99720 1/20 0.52
S1PR1 P21453 1/20 0.51
S1PR5 Q9H228 1/20 0.51
GRIN2B Q13224 1/20 0.51
GBA1 P04062 1/20 0.50
ALDH1A1 P00352 1/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19680503 0.86 ALDH1A1 (0.55) FUCA1SIGMAR1ALDH1A1KDM4E
SCHEMBL19689038 0.86 ALDH1A1 (0.55) FUCA1SIGMAR1ALDH1A1KDM4E
SCHEMBL8948752 0.82 S1PR5 (0.54) FUCA1SIGMAR1S1PR1S1PR5GRIN2B
SCHEMBL19450643 0.81 ACHE (0.61) SIGMAR1KDM4E
SCHEMBL16544830 0.81 FUCA1 (0.55) FUCA1SIGMAR1S1PR1S1PR5GBA1
SCHEMBL1860555 0.78 FUCA1 (1.00) FUCA1SIGMAR1S1PR1S1PR5GBA1
SCHEMBL7637770 0.78 FUCA1 (1.00) FUCA1SIGMAR1S1PR1S1PR5GBA1
SCHEMBL7637709 0.78 FUCA1 (1.00) FUCA1SIGMAR1S1PR1S1PR5GBA1
SCHEMBL84802 0.78 FUCA1 (0.85) FUCA1SIGMAR1S1PR1S1PR5GRIN2B
SCHEMBL71063 0.78 FUCA1 (0.85) FUCA1SIGMAR1S1PR1S1PR5GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3253752-B1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2023-08-16 EP disclosed
EP-0165636-B1 PROCESS FOR PREPARING AZETIDINE DERIVATIVES AND INTERMEDIATES THEREIN SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1988-08-10 EP disclosed
EP-0165636-A1 Process for preparing azetidine derivatives and intermediates therein SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1985-12-27 EP disclosed