SCHEMBL10652373

SCHEMBL10652373

COc1ccc2c(c1)c1oc(-c3nnn[nH]3)c(OC)c1n2-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
MAPT P10636 3/20 0.39
HTT P42858 2/20 0.39
EDNRA P25101 2/20 0.35
ALDH1A1 P00352 5/20 0.35
HPGD P15428 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
FGFR1 P11362 1/20 0.34
HSD17B10 Q99714 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR6 P50406 1/20 0.34
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
PLA2G2A P14555 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10652614 0.89 LMNA (0.41) KDM4EALDH1A1MEN1KMT2AHSD17B10
SCHEMBL10652305 0.78 KDM4E (0.41) KDM4EMAPTHTTEDNRAALDH1A1
SCHEMBL10652379 0.78 PPARG (0.33) KDM4EMAPTALDH1A1HPGDMEN1
SCHEMBL10653000 0.76 KDM4E (0.45) KDM4EMAPTHTTEDNRAALDH1A1
SCHEMBL10655975 0.76 KDM4E (0.45) KDM4EMAPTHTTEDNRAALDH1A1
SCHEMBL10652350 0.76 KDM4E (0.56) KDM4EMAPTHTTEDNRAALDH1A1
SCHEMBL10655784 0.75 PABPC1 (0.38) KDM4EMAPTHTTALDH1A1HPGD
SCHEMBL10654966 0.73 KMT2A (0.40) KDM4EMAPTHTTEDNRAALDH1A1
SCHEMBL10373185 0.73 ALDH1A1 (0.45) KDM4EMAPTHTTALDH1A1HPGD
SCHEMBL10655257 0.72 KDM4E (0.51) KDM4EMAPTHTTEDNRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0092380-B1 ANTIALLERGIC 4H-FURO(3,2-B)INDOLES AND THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1988-01-20 EP claimed
US-4596814-A Antiallergens WARNER-LAMBERT COMPANY (US) 1986-06-24 US claimed
EP-0092380-A2 Antiallergic 4H-furo(3,2-b)indoles and their production WARNER-LAMBERT COMPANY (US) 1983-10-26 EP claimed
EP-0092380-B1 ANTIALLERGIC 4H-FURO(3,2-B)INDOLES AND THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1988-01-20 EP disclosed
US-4596814-A Antiallergens WARNER-LAMBERT COMPANY (US) 1986-06-24 US disclosed
US-4503236-A Antiallergic 4Hfuro[3,2-b]indoles WARNER-LAMBERT COMPANY (US) 1985-03-05 US disclosed
EP-0092380-A2 Antiallergic 4H-furo(3,2-b)indoles and their production WARNER-LAMBERT COMPANY (US) 1983-10-26 EP disclosed