SCHEMBL10654412

SCHEMBL10654412

CCOc1c(C(N)=O)oc2c3ccccc3n(-c3ccccc3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.41
MAPT P10636 3/20 0.40
HPGD P15428 3/20 0.40
LMNA P02545 2/20 0.40
MAPK10 P53779 2/20 0.40
PPARG P37231 1/20 0.40
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
PLA2G2A P14555 1/20 0.40
ALDH1A1 P00352 7/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 3/20 0.38
HSD17B10 Q99714 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGER4 P35408 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 3/20 0.37
POLB P06746 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10654421 0.91 ALDH1A1 (0.44) RECQLMAPTHPGDPPARGPLA2G2A
SCHEMBL10652918 0.88 MAPK8 (0.43) RECQLMAPTHPGDPPARGALOX15
SCHEMBL10654374 0.87 LMNA (0.42) RECQLMAPTHPGDLMNAALOX15
SCHEMBL10654464 0.78 RECQL (0.35) RECQLMAPTHPGDLMNAMAPK10
SCHEMBL10654988 0.78 MEN1 (0.52) MAPTHPGDPPARGTP53ALDH1A1
SCHEMBL10653794 0.77 LMNA (0.43) RECQLMAPTHPGDLMNAPPARG
SCHEMBL10654499 0.77 RECQL (0.36) RECQLMAPTHPGDPPARGTP53
SCHEMBL10654396 0.77 ALDH1A1 (0.38) RECQLMAPTHPGDLMNAPPARG
SCHEMBL10654418 0.76 MEN1 (0.48) MAPTHPGDTP53ALOX15ALDH1A1
SCHEMBL10654033 0.76 KDM4E (0.51) MAPTHPGDLMNATP53PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0092380-B1 ANTIALLERGIC 4H-FURO(3,2-B)INDOLES AND THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1988-01-20 EP disclosed
US-4596814-A Antiallergens WARNER-LAMBERT COMPANY (US) 1986-06-24 US disclosed
US-4503236-A Antiallergic 4Hfuro[3,2-b]indoles WARNER-LAMBERT COMPANY (US) 1985-03-05 US disclosed
EP-0092380-A2 Antiallergic 4H-furo(3,2-b)indoles and their production WARNER-LAMBERT COMPANY (US) 1983-10-26 EP disclosed