SCHEMBL10654584

SCHEMBL10654584

CCOC(=O)C1CN(C(=O)OCC)CCC1=O

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
ALDH1A1 P00352 8/20 0.42
LMNA P02545 1/20 0.41
GAA P10253 3/20 0.41
KDM4E B2RXH2 3/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethylene SCHEMBL10653813 0.97 MAPT (0.43) MAPTALDH1A1LMNAGAAKDM4E
SCHEMBL10654314 0.93 MAPT (0.43) MAPTALDH1A1LMNAGAAKDM4E
SCHEMBL31454859 0.91 ALDH1A1 (0.42) MAPTALDH1A1LMNAGAAKDM4E
SCHEMBL533925 0.91 LMNA (0.45) MAPTALDH1A1LMNAGAAKDM4E
Ethylene SCHEMBL10844325 0.90 MAPT (0.41) MAPTALDH1A1LMNAGAAKDM4E
SCHEMBL5871351 0.89 MAPT (0.44) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL2127522 0.89 MAPT (0.44) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL29450286 0.89 MAPT (0.46) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL183637 0.89 MAPT (0.46) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL9310424 0.88 MAPT (0.38) MAPTALDH1A1LMNAGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126654-B1 TETRAHYDROISOXAZOLO(4,5-C)PYRIDINE DERIVATIVES AND PREPARATION THEREOF H. LUNDBECK A/S (DK) 1988-05-04 EP disclosed
US-4608378-A Tetrahydroisoxazolo[4,5-c]pyridine derivatives useful in the treatment of malfunctions of the acetylcholine or muscarinic systems H. LUNDBECK A/S (DK) 1986-08-26 US disclosed
EP-0126654-A1 Tetrahydroisoxazolo(4,5-c)pyridine derivatives and preparation thereof H. LUNDBECK A/S (DK) 1984-11-28 EP disclosed