SCHEMBL10656103

SCHEMBL10656103

COc1ccc(-c2csc(SC)c2C#N)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
MAPT P10636 5/20 0.52
KDM4E B2RXH2 4/20 0.52
HPGD P15428 3/20 0.52
NPSR1 Q6W5P4 3/20 0.52
RXFP1 Q9HBX9 2/20 0.52
PTPN1 P18031 2/20 0.47
PRKCZ Q05513 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
GAA P10253 1/20 0.43
ADORA1 P30542 2/20 0.42
SQOR Q9Y6N5 1/20 0.42
PIM1 P11309 4/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10656806 0.83 NPSR1 (0.42) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL10651575 0.82 PDCD1 (0.46) ALDH1A1MAPTKDM4ENPSR1RXFP1
SCHEMBL10655134 0.82 KDM4E (0.43) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL10655060 0.81 GRIA4 (0.47) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL13991789 0.80 PRKCZ (0.47) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL10654580 0.79 CYP2A6 (0.40) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL15629589 0.79 PRKCZ (0.68) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL10653315 0.78 KIF11 (0.42) ALDH1A1MAPTKDM4ERXFP1PTPN1
SCHEMBL10656293 0.75 PRKCZ (0.43) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL10651211 0.75 MAPK14 (0.40) ALDH1A1MAPTPRKCZADORA1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273602-A1 3-Cyano-4-arylthiophenes ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed