SCHEMBL10656262

SCHEMBL10656262

CCc1ccc(N)c(C(O)=S)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
CDC25B P30305 1/20 0.47
CASP6 P55212 1/20 0.47
RCE1 Q9Y256 1/20 0.47
KDM4E B2RXH2 3/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
TRPA1 O75762 1/20 0.41
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10659876 0.85 ALDH1A1 (0.44) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL11165456 0.82 SKP2 (0.57) ALDH1A1CDC25BCASP6RCE1HPGD
SCHEMBL10660025 0.81 SKP2 (0.51) ALDH1A1KDM4EHSD17B10SKP2
SCHEMBL648210 0.81 ALDH1A1 (0.72) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL11387602 0.79 ALDH1A1 (0.45) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL20670595 0.77 ALDH1A1 (0.54) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL4097033 0.77 ALDH1A1 (0.54) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL10655549 0.77 XDH (0.46) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL24629784 0.76 ALDH1A1 (0.45) ALDH1A1CDC25BCASP6RCE1KDM4E
SCHEMBL9041416 0.76 ALDH1A1 (0.53) ALDH1A1CDC25BCASP6RCE1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4745116-A INHIBITORS OF SERINE PROTEASE SYNTEX (U.S.A.) INC. (US) 1988-05-17 US disclosed
US-4665070-A SERINE PROTEINASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1987-05-12 US disclosed
EP-0206323-A1 2-Oxy-4H-3,1-benzoxazin-4-one derivatives and related compounds SYNTEX (U.S.A.) INC. (US) 1986-12-30 EP disclosed