SCHEMBL10658912

SCHEMBL10658912

O=C(c1ccoc1)c1ccc(O)c(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HTT P42858 1/20 0.40
MMP2 P08253 1/20 0.36
CYP3A4 P08684 2/20 0.35
HDAC1 Q13547 1/20 0.35
TRPA1 O75762 1/20 0.35
CNR2 P34972 1/20 0.35
MAPT P10636 2/20 0.34
PTPN1 P18031 1/20 0.33
PTPN6 P29350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14419533 0.79 CA1 (0.51) MAPK1ALDH1A1MEN1LMNAPKM
SCHEMBL10662982 0.78 MAPT (0.43) MAPK1ALDH1A1MEN1LMNAHPGD
SCHEMBL11055051 0.78 MAPK1 (0.50) MAPK1ALDH1A1MEN1LMNAPKM
SCHEMBL10455760 0.75 LMNA (0.58) MAPK1ALDH1A1MEN1LMNAPKM
SCHEMBL11336100 0.75 MAPK1 (0.53) MAPK1ALDH1A1MEN1LMNAPKM
SCHEMBL8866037 0.73 TRPA1 (0.48) ALDH1A1MEN1HPGDKMT2ACYP3A4
SCHEMBL10661164 0.72 HTT (0.60) ALDH1A1MEN1LMNAHPGDKMT2A
SCHEMBL10660598 0.72 KCNMA1 (0.43) MAPK1ALDH1A1MEN1LMNAPKM
SCHEMBL10662231 0.71 SRD5A2 (0.51) MAPK1ALDH1A1MEN1PKMHPGD
SCHEMBL11256540 0.69 RAB9A (0.59) MAPK1ALDH1A1MEN1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4728662-A DIURETICS, URICOSURICS, HYPOTENSIVES HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-03-01 US disclosed
US-4673746-A DIURETICS, HYPOTENSIVES HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1987-06-16 US disclosed
EP-0002666-B1 1,2-BENZISOXAZOLYLOXY (OR THIO) ACETIC ACIDS AND RELATED COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-02-17 EP disclosed