SCHEMBL10659508

SCHEMBL10659508

Cc1ccc(C)c(C(=O)OC(C)C)c1NS(=O)(=O)c1nc2ncccn2n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.46
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 2/20 0.37
THRB P10828 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RAB9A P51151 1/20 0.35
TP53 P04637 1/20 0.35
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
CRHBP P24387 1/20 0.33
HTT P42858 1/20 0.33
CRHR2 Q13324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10666392 0.90 HPGD (0.43) LMNAHPGDSMN1; SMN2ALDH1A1THRB
SCHEMBL10664496 0.88 HPGD (0.43) LMNAHPGDSMN1; SMN2ALDH1A1THRB
SCHEMBL10664350 0.87 HPGD (0.47) LMNAHPGDSMN1; SMN2ALDH1A1THRB
SCHEMBL10664174 0.87 THRB (0.44) LMNAHPGDSMN1; SMN2ALDH1A1THRB
SCHEMBL10666055 0.87 HPGD (0.44) LMNAHPGDSMN1; SMN2ALDH1A1THRB
SCHEMBL9831039 0.86 ALDH1A1 (0.33) LMNAALDH1A1TP53MAPTGAA
SCHEMBL9833022 0.84 MAPT (0.33) LMNAHPGDALDH1A1HSD17B10TP53
SCHEMBL9831000 0.84 L3MBTL1 (0.41) LMNASMN1; SMN2ALDH1A1RAB9AMEN1
SCHEMBL10665699 0.81 LMNA (0.42) LMNAHPGDSMN1; SMN2THRBHSD17B10
SCHEMBL10660546 0.81 HPGD (0.40) LMNAHPGDSMN1; SMN2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed