SCHEMBL10668372

SCHEMBL10668372

CC1=C(C(=O)OCC2CCCO2)C(c2cccc([N+](=O)[O-])c2)C(C(=O)OC2CC(C)CC(C)(C)C2)=C(C)N1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.55
KMT2A Q03164 3/20 0.55
CACNA1C Q13936 8/20 0.54
CACNA1F O60840 7/20 0.54
CACNA1D Q01668 7/20 0.54
CACNA1S Q13698 7/20 0.54
ADORA3 P0DMS8 2/20 0.54
HIF1A Q16665 3/20 0.51
MEN1 O00255 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
MAPT P10636 2/20 0.51
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
GPR55 Q9Y2T6 1/20 0.51
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955134 0.88 POLB (0.68) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10665954 0.87 CACNA1F (0.72) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL7416441 0.85 POLB (0.64) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL7132512 0.85 POLB (0.75) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10667044 0.83 HIF1A (0.64) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10668367 0.81 CACNA1C (0.49) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10670264 0.78 KMT2A (0.76) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10666490 0.77 CACNA1F (0.57) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL10900830 0.76 MEN1 (0.76) POLBKMT2ACACNA1CCACNA1FCACNA1D
SCHEMBL11063168 0.76 CACNA1F (0.79) POLBKMT2ACACNA1CCACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4656181-A CARDIOTONIC AGENTS CERMOL S.A. (CH) 1987-04-07 US claimed
US-4727066-A CARDIOVASCULAR DISORDERS CERMOL S.A. (CH) 1988-02-23 US disclosed
US-4656181-A CARDIOTONIC AGENTS CERMOL S.A. (CH) 1987-04-07 US disclosed