SCHEMBL1067286

SCHEMBL1067286

CC(C)(F)COS(=O)(=O)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.36
CA1 P00915 2/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11612358 0.85 CA2 (0.40) CA2CA1CA9
SCHEMBL21312124 0.85 CA1 (0.36) CA2CA1CA9
SCHEMBL4813050 0.85 CA2 (0.36) CA2CA1CA9
SCHEMBL3242894 0.85 CA2 (0.36) CA2CA1CA9
SCHEMBL20602111 0.81 CA2 (0.34) CA2CA1CA9
SCHEMBL18896075 0.81 CA2 (0.34) CA2CA1CA9
SCHEMBL17858943 0.79 CA2 (0.33) CA2CA1CA9
SCHEMBL3241936 0.79 CA2 (0.33) CA2CA1CA9
SCHEMBL1855129 0.79 CA2 (0.39) CA2CA1CA9
SCHEMBL26912 0.79 CA2 (0.56) CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 283 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11672785-B2 Tetrahydro-1H-pyrido [3,4-b]indole anti-estrogenic drugs OLEMA PHARMACEUTICALS, INC. (US) 2023-06-13 US claimed
US-20220370421-A1 TETRAHYDRO-1H-PYRIDO [3,4-b]INDOLE ANTI-ESTROGENIC DRUGS OLEMA PHARMACEUTICALS, INC. 2022-11-24 US claimed
US-20260144778-A1 REGIMENS OF ESTROGEN RECEPTOR ANTAGONISTS OLEMA PHARMACEUTICALS, INC. (US) 2026-05-28 US disclosed
EP-4736854-A2 HETEROCYCLIC COMPOUNDS AS MODULATORS OF BCL6 AS LIGAND DIRECTED DEGRADERS Bristol-Myers Squibb Company (US) 2026-05-06 EP disclosed
US-12606541-B2 PPARg modulators and methods of use EISAI R&D MANAGEMENT CO., LTD. (JP) 2026-04-21 US disclosed
US-20260103461-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF OLEMA PHARMACEUTICALS INC (US) 2026-04-16 US disclosed
EP-4514473-B1 HETEROCYCLIC COMPOUNDS AS MODULATORS OF BCL6 AS LIGAND DIRECTED DEGRADERS BRISTOL MYERS SQUIBB CO (US) 2026-02-18 EP disclosed
US-20260028341-A1 IMIDAZOTRIAZINE DERIVATIVES AS IL-17 MODULATORS UCB Biopharma SRL (BE) 2026-01-29 US disclosed
US-20260007681-A1 INDOLE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS UNIV MICHIGAN (US) 2026-01-08 US disclosed
US-20250368625-A1 PIPERAZINES Grünenthal GmbH (DE) 2025-12-04 US disclosed
US-20250320183-A1 Modulators of BCL6 as Ligand Directed Degraders CELGENE CORPORATION (US) 2025-10-16 US disclosed
US-20100087429-A1 SPIRO-TRICYCLIC RING COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2010-04-08 US disclosed
WO-2010030954-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETASECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2010-03-18 WO disclosed
US-20090264445-A1 PYRROLIDINONE GLUCOKINASE ACTIVATORS BERTHEL STEVEN JOSEPH 2009-10-22 US disclosed
WO-2009127546-A1 PYRROLIDINONE GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2009-10-22 WO disclosed
EP-2091928-A2 3-(2-ACYLAMINO-1-HYDROXYETHYL)- MORPHOLINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2009-08-26 EP disclosed
US-7429674-B2 Process for preparing fluoroleucine alkyl esters MERCK & CO. INC.. (US) 2008-09-30 US disclosed
US-7429674-B2 Process for preparing fluoroleucine alkyl esters MERCK & CO. INC.. (US) 2008-09-30 US disclosed
US-20070225267-A1 3-(2-Acylamino-1-Hydroxyethyl)-Morpholine Derivatives and Their Use as Bace Inhibitors ELI LILLY AND COMPANY 2007-09-27 US disclosed
WO-2006034093-A2 3- (2-ACYLAMINO-1-HYDROXYETHYL)- MORPHOLINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS ELLI LILLY AND COMPANY (US) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11672785-B2 Tetrahydro-1H-pyrido [3,4-b]indole anti-estrogenic drugs ESR1, CYP19A1, HSD17B11 CA2 1896/4885CA1 1198/4885CA9 3028/4885
US-20260103461-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ESRRA, GPER1, ESR2 CA2 699/4885CA1 745/4885CA9 1354/4885
US-20070225267-A1 3-(2-Acylamino-1-Hydroxyethyl)-Morpholine Derivatives and Their Use as Bace Inhibitors BACE1, BACE2, APP CA2 2660/4885CA1 1464/4885CA9 3327/4885
US-20090264445-A1 PYRROLIDINONE GLUCOKINASE ACTIVATORS GCKR, GCK, PDK2 CA2 2535/4885CA1 4305/4885CA9 2829/4885
US-20260028341-A1 IMIDAZOTRIAZINE DERIVATIVES AS IL-17 MODULATORS IL17A, IL6ST, IL6 CA2 1939/4885CA1 2509/4885CA9 3345/4885
US-20260007681-A1 INDOLE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS ESRRA, ESR2, AR CA2 871/4885CA1 1137/4885CA9 772/4885
US-20250320183-A1 Modulators of BCL6 as Ligand Directed Degraders BCL6, BCL6B, BCL3 CA2 4634/4885CA1 3464/4885CA9 3422/4885
US-12606541-B2 PPARg modulators and methods of use PPARG, PPARA, PPARD CA2 2393/4885CA1 4704/4885CA9 3899/4885
US-20100087429-A1 SPIRO-TRICYCLIC RING COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE BACE1, BACE2, APP CA2 2229/4885CA1 85/4885CA9 3008/4885
US-20250368625-A1 PIPERAZINES SSTR4, SSTR5, SSTR2 CA2 1871/4885CA1 3396/4885CA9 3944/4885
US-20220370421-A1 TETRAHYDRO-1H-PYRIDO [3,4-b]INDOLE ANTI-ESTROGENIC DRUGS ESR1, CYP19A1, HSD17B11 CA2 1896/4885CA1 1198/4885CA9 3028/4885
US-20260144778-A1 REGIMENS OF ESTROGEN RECEPTOR ANTAGONISTS ESR1, ESR2, PGR CA2 2973/4885CA1 4038/4885CA9 3077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.