SCHEMBL10679358

SCHEMBL10679358

CN1CCCC(COc2cccc3oc(-c4ccccc4)cc(=O)c23)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.59
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 3/20 0.57
AR P10275 3/20 0.57
CYP3A4 P08684 3/20 0.57
TP53 P04637 2/20 0.57
HSD17B10 Q99714 2/20 0.57
MAPT P10636 2/20 0.57
HPGD P15428 2/20 0.57
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10682290 0.82 MAOA (0.67) SIGMAR1BCHEACHEMAOAMAOB
SCHEMBL10681862 0.81 SIGMAR1 (0.61) SIGMAR1ALDH1A1KDM4EMAPTMAOA
SCHEMBL10682513 0.81 ALDH1A1 (0.53) SIGMAR1ALDH1A1KDM4EARCYP3A4
SCHEMBL10684580 0.81 SIGMAR1 (0.52) SIGMAR1ALDH1A1KDM4EARCYP3A4
SCHEMBL7370312 0.80 HPGD (0.49) ALDH1A1KDM4EARCYP3A4TP53
SCHEMBL10682405 0.80 ALDH1A1 (0.56) SIGMAR1ALDH1A1KDM4EARCYP3A4
SCHEMBL10682530 0.79 CHRNB2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL10677213 0.78 SIGMAR1 (0.62) SIGMAR1ALDH1A1KDM4EARCYP3A4
SCHEMBL9205310 0.77 AR (0.61) SIGMAR1ALDH1A1KDM4EARCYP3A4
SCHEMBL9137293 0.75 ALDH1A1 (0.72) SIGMAR1ALDH1A1KDM4EARCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed