SCHEMBL10686705

SCHEMBL10686705

CC(Cc1cccc(Br)c1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.50
SIGMAR1 Q99720 1/20 0.49
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
PLA2G10 O15496 3/20 0.47
PLA2G2A P14555 3/20 0.47
PLA2G1B P04054 1/20 0.47
PLA2G5 P39877 1/20 0.47
PLA2G2C Q5R387 1/20 0.47
PLA2G12B Q9BX93 1/20 0.47
PLA2G12A Q9BZM1 1/20 0.47
PLA2G2F Q9BZM2 1/20 0.47
PLA2G3 Q9NZ20 1/20 0.47
PLA2G2E Q9NZK7 1/20 0.47
PLA2G2D Q9UNK4 1/20 0.47
TBXAS1 P24557 2/20 0.47
FFAR1 O14842 2/20 0.45
HCAR2 Q8TDS4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14870372 1.00 PTGES (0.50) PTGESSIGMAR1MEN1NPC1RAB9A
SCHEMBL31189307 1.00 PTGES (0.50) PTGESSIGMAR1MEN1NPC1RAB9A
SCHEMBL8257100 0.87 TBXAS1 (0.53) PLA2G10PLA2G2APLA2G1BPLA2G5PLA2G2C
SCHEMBL3471743 0.84 HCAR2 (0.47) PTGESSIGMAR1NPC1RAB9AFFAR1
SCHEMBL25173384 0.83 TSHR (0.51) PTGESSIGMAR1MEN1NPC1RAB9A
SCHEMBL6029226 0.83 FFAR1 (0.67) FFAR1MAOB
SCHEMBL1124990 0.83 PLA2G10 (0.47) MEN1NPC1RAB9AKMT2APLA2G10
SCHEMBL27785183 0.82 HCAR2 (0.46) PTGESSIGMAR1NPC1RAB9AFFAR1
SCHEMBL18367812 0.82 ALDH1A1 (0.49) PTGESSIGMAR1MEN1NPC1RAB9A
SCHEMBL27641743 0.82 ALDH1A1 (0.49) PTGESSIGMAR1MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112930347-A Inhibitors of KEAP1-Nrf2 protein-protein interactions 詹森药业有限公司 2021-06-08 CN disclosed
US-4738803-A ENZYME INHIBITORS ROQUES BERNARD (FR) 1988-04-19 US disclosed
US-4618708-A ENKEPHALINASE INHIBITOR, ANALGESICS, ANTIDEPRESSANT, ANTIDIARRHEA, OR HYPOTENSIVE AGENT ROQUES BERNARD (FR) 1986-10-21 US disclosed