SCHEMBL10690630

SCHEMBL10690630

Cc1sc(-c2ccccc2)c(-c2ccccc2)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.41
GRM6 O15303 4/20 0.41
CHEK1 O14757 1/20 0.39
AKT2 P31751 1/20 0.39
LIMK1 P53667 1/20 0.38
MAPT P10636 3/20 0.37
HTT P42858 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37
KMT2A Q03164 1/20 0.37
RELA Q04206 1/20 0.37
GRM5 P41594 1/20 0.37
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10109209 0.84 ALOX5 (0.42) ALOX5GRM6CHEK1AKT2MAPT
SCHEMBL13713793 0.82 GRM6 (0.47) ALOX5GRM6LIMK1MAPTHTT
SCHEMBL13093559 0.82 CHEK1 (0.42) CHEK1AKT2MAPTHTTALDH1A1
SCHEMBL26724795 0.77 ALOX5 (0.40) ALOX5GRM6CHEK1AKT2LIMK1
SCHEMBL21494935 0.77 GRM6 (0.49) ALOX5GRM6LIMK1MAPTHTT
SCHEMBL1224397 0.76 MAPT (0.56) ALOX5GRM6CHEK1AKT2MAPT
SCHEMBL12262883 0.74 ALOX5 (0.51) ALOX5GRM6CHEK1AKT2MAPT
SCHEMBL13337266 0.74 AKT2 (0.46) ALOX5CHEK1AKT2MAPTHTT
SCHEMBL16996824 0.74 GRM6 (0.52) ALOX5GRM6LIMK1MAPTHTT
SCHEMBL10698380 0.72 ALOX5 (0.48) ALOX5GRM6LIMK1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4749712-A Antiinflammatory and/or analgesic 5-alkylthiophenes E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-06-07 US disclosed