SCHEMBL10691177

SCHEMBL10691177

Clc1ccc(-n2ccnc2CC2=CCCC=C2)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.36
GRM5 P41594 9/20 0.34
HCAR1 Q9BXC0 1/20 0.33
PHGDH O43175 2/20 0.32
CYP11B2 P19099 1/20 0.32
NOTUM Q6P988 1/20 0.32
OPRL1 P41146 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
AKR1C3 P42330 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690683 0.79 TSHR (0.43) KCNH2LMNAHTT
SCHEMBL31376140 0.71 TLR8 (0.50) KCNH2GRM5HCAR1NOTUM
SCHEMBL28240610 0.70 KCNH2 (0.38) KCNH2GRM5HCAR1CYP11B2NOTUM
SCHEMBL8047156 0.66 HCAR1 (0.42) KCNH2HCAR1CYP11B2NOTUMLMNA
SCHEMBL4959137 0.64 LMNA (0.38) KCNH2GRM5HCAR1CYP11B2LMNA
SCHEMBL10691328 0.62 POLB (0.41)
SCHEMBL28197166 0.61 CYP2D6 (0.43) KCNH2HCAR1CYP11B2LMNA
SCHEMBL5173711 0.60 IDO1 (0.49) KCNH2HCAR1CYP11B2NOTUMLMNA
SCHEMBL7633090 0.60
Hydrochloric Acid SCHEMBL11260141 0.59 KCNH2 (0.39) KCNH2GRM5HCAR1CYP11B2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4732989-A INTERMEDIATES FOR BACTERICIDES G. D. SEARLE & CO. (US) 1988-03-22 US disclosed
US-4661602-A ANTIANAEROBIC AGENTS G. D. SEARLE & CO. (US) 1987-04-28 US disclosed