SCHEMBL10692459

SCHEMBL10692459

COC(=O)CC[C@H](NC(=O)c1ccc(N(C)C(=O)OCc2ccccc2)cc1)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
RAB9A P51151 2/20 0.47
GAA P10253 1/20 0.47
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
ABCB1 P08183 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ACE P12821 1/20 0.43
MAPK14 Q16539 1/20 0.42
KYNU Q16719 1/20 0.41
LMNA P02545 1/20 0.41
GLA P06280 1/20 0.41
ALOX5 P09917 1/20 0.41
CCKBR P32239 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19918328 0.87 CYP26A1 (0.42) CA1CA2RAB9AGAAALDH1A1
SCHEMBL19899438 0.86 FOLH1 (0.50) CA1CA2LMNA
SCHEMBL19899429 0.86 FOLH1 (0.50) CA1CA2LMNA
SCHEMBL8973061 0.83 RAB9A (0.61) CA1CA2RAB9AGAAALDH1A1
SCHEMBL19918338 0.82 CA1 (0.54) CA1CA2RAB9AGAAMAPT
SCHEMBL27660162 0.82 ALOX5 (0.52) CA1CA2RAB9AGAAALDH1A1
SCHEMBL27660160 0.82 ALOX5 (0.52) CA1CA2RAB9AGAAALDH1A1
SCHEMBL10692464 0.81 CA1 (0.48) CA1CA2RAB9AGAAALDH1A1
SCHEMBL13668076 0.80 CA1 (0.51) CA1CA2RAB9AGAAALDH1A1
SCHEMBL7087075 0.78 KYNU (0.59) ALDH1A1KYNU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4725687-A ANTITUMOR AGENTS; SIDE EFFECT REDUCTION; POTENCY SOUTHERN RESEARCH INSTITUTE (US) 1988-02-16 US disclosed