SCHEMBL10695000

SCHEMBL10695000

COc1ccc(CCN(C)C(=O)CCC2Cc3cc(OC)c(OC)cc3C2=O)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
ACHE P22303 5/20 0.53
TDP1 Q9NUW8 1/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10427929 0.90 CDK8 (0.53) CDK8CLK4ACHETDP1NPC1
SCHEMBL10693928 0.84 LTB4R (0.53) ACHE
SCHEMBL10696013 0.84 CYP3A4 (0.56) ACHECYP1A2CYP3A4CYP2D6
SCHEMBL10427950 0.81 DRD2 (0.44) CDK8CLK4ACHE
SCHEMBL10699939 0.78 ACHE (0.49) CDK8CLK4ACHETDP1MEN1
SCHEMBL10426976 0.76 ACHE (0.54) ACHE
SCHEMBL10696001 0.76 ACHE (0.51) ACHE
SCHEMBL10427884 0.76 LTB4R (0.52) ACHEMEN1KMT2A
SCHEMBL10427190 0.75 ACHE (0.52) ACHEKMT2A
SCHEMBL10427932 0.75 LTB4R (0.52) ACHECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259782-A1 Naphthalene and indane derivatives, medicaments containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1988-03-16 EP disclosed