SCHEMBL10695089

SCHEMBL10695089

c1cc2c(cc1C1CO1)CCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.41
GSTO1 P78417 2/20 0.39
ALDH1A1 P00352 2/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
PARP1 P09874 1/20 0.37
HPGD P15428 2/20 0.36
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MGLL Q99685 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
BLM P54132 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10689892 0.96 TSHR (0.41) TSHRGSTO1ALDH1A1CA12CA1
SCHEMBL10386376 0.76 HPGD (0.33) ALDH1A1CA12CA1CA2CA7
SCHEMBL31290248 0.74 ALDH1A1 (0.41) ALDH1A1CA12CA1CA2CA7
SCHEMBL10386635 0.72 ADRA2A (0.31) HPGDADRA2AADRA2BADRA2C
SCHEMBL46155 0.71 TSHR (0.72) TSHRGSTO1PARP1ADRA2A
SCHEMBL10879536 0.71 EPHX2 (0.49) ALDH1A1CA12CA1CA2CA7
SCHEMBL18649887 0.70 LTA4H (0.54) TSHRALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL8941787 0.69 TSHR (0.45) TSHRALDH1A1PARP1HPGDNPC1
SCHEMBL12971972 0.69 KDM1A (0.46) ADRA2ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL16430852 0.68 TSHR (0.35) TSHRGSTO1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4751222-A 2,3,4,5-tetrahydro-1H-3-benzazepines and CNS affecting use thereof NOVO INDUSTRI A/S (DK) 1988-06-14 US disclosed
EP-0200455-A2 2,3,4,5-tetrahydro-1H-3-benzazepines substituted in position 5 NOVO NORDISK A/S (DK) 1986-11-05 EP disclosed