SCHEMBL10695581

SCHEMBL10695581

O=C(CCCc1ccccc1)Cc1cccnc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 10/20 0.60
NAPRT Q6XQN6 1/20 0.60
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 1/20 0.55
EPHX2 P34913 1/20 0.52
KMT2A Q03164 1/20 0.52
HDAC3 O15379 1/20 0.51
MAPK1 P28482 1/20 0.51
ADRA1A P35348 1/20 0.51
HDAC4 P56524 1/20 0.51
SLC6A3 Q01959 1/20 0.51
HDAC1 Q13547 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695569 0.85 MEN1 (0.50) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL10695456 0.85 KMT2A (0.53) TBXAS1KMT2ASMN1; SMN2
SCHEMBL7362509 0.83 NAPRT (0.72) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL8664876 0.83 HDAC1 (0.67) HDAC3MAPK1ADRA1AHDAC4SLC6A3
SCHEMBL1538161 0.83 NAPRT (0.57) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL3253168 0.81 NAPRT (0.74) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL28975712 0.80 NAPRT (0.62) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL30612524 0.80 TBXAS1 (0.90) TBXAS1NAPRTHDAC3MAPK1ADRA1A
SCHEMBL30195679 0.80 NAPRT (0.62) TBXAS1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL1583762 0.80 TBXAS1 (0.90) TBXAS1NAPRTHDAC3MAPK1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267439-A2 Alpha-(phenylalkyl) pyridinealkanol derivatives G.D. Searle & Co. (US) 1988-05-18 EP disclosed