SCHEMBL10695768

SCHEMBL10695768

COc1nccnc1Nc1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
CA2 P00918 8/20 0.57
CA9 Q16790 8/20 0.57
CA1 P00915 7/20 0.57
CA12 O43570 5/20 0.57
MAPT P10636 1/20 0.52
GAA P10253 1/20 0.50
IKBKB O14920 1/20 0.49
EGFR P00533 4/20 0.48
KDR P35968 3/20 0.48
ENPP3 O14638 2/20 0.47
ERBB3 P21860 2/20 0.47
CA14 Q9ULX7 3/20 0.47
POLB P06746 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CA6 P23280 2/20 0.47
CA5A P35218 2/20 0.47
CA7 P43166 2/20 0.47
ROCK1 Q13464 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfalene SCHEMBL28086248 0.81 MEN1 (0.90) MEN1KMT2ACA2CA9CA1
SCHEMBL7052503 0.79 ESR1 (0.61) CA2CA9CA1CA12EGFR
SCHEMBL26656469 0.76 CA1 (0.47) CA2CA9CA1CA12IKBKB
Sulfalene SCHEMBL28404 0.73 MEN1 (1.00) MEN1KMT2AMAPTGAAALDH1A1
Sulfalene SCHEMBL1893333 0.73 MEN1 (1.00) MEN1KMT2AMAPTGAAALDH1A1
Sulfanilamide SCHEMBL27917543 0.73 KMT2A (0.55) MEN1KMT2ACA2CA9CA1
SCHEMBL28747203 0.73 CA1 (0.67) MEN1KMT2ACA2CA9CA1
SCHEMBL24477607 0.72 CA2 (0.59) CA2CA9CA1CA12IKBKB
SCHEMBL24477734 0.72 CDK2 (0.60) CA2CA9CA1CA12IKBKB
SCHEMBL27962184 0.72 CA1 (0.62) CA2CA9CA1CA12EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255100-A2 Use of trimetrexate and its salts for the preparation of pharmaceutical compositions for treating infections of the mycobacterium-avium-intracellulare complex WARNER-LAMBERT COMPANY (US) 1988-02-03 EP claimed