SCHEMBL10696939

SCHEMBL10696939

CCCCCN1C(=O)C(C)(C)c2cc(NC(=O)c3ccco3)c([N+](=O)[O-])cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.49
RAB9A P51151 6/20 0.49
KMT2A Q03164 6/20 0.49
NPC1 O15118 4/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
ALDH1A1 P00352 7/20 0.49
PKM P14618 1/20 0.43
MEN1 O00255 4/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
POLB P06746 3/20 0.41
TSHR P16473 2/20 0.41
MAPT P10636 5/20 0.40
MITF O75030 1/20 0.40
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10703903 0.94 SMN1; SMN2 (0.52) SMN1; SMN2RAB9AKMT2ANPC1NFKB1
SCHEMBL10714503 0.90 ALDH1A1 (0.53) SMN1; SMN2RAB9AKMT2ANPC1NFKB1
SCHEMBL10696545 0.84 LMNA (0.38) SMN1; SMN2RAB9AKMT2ANPC1ALDH1A1
SCHEMBL2490357 0.83 MAPT (0.56) RAB9AKMT2ANPC1ALDH1A1PKM
SCHEMBL10699652 0.83 NPC1 (0.49) SMN1; SMN2RAB9AKMT2ANPC1ALDH1A1
SCHEMBL10700893 0.83 SETD7 (0.41) SMN1; SMN2RAB9AKMT2ANPC1ALDH1A1
SCHEMBL10698960 0.82 MAPT (0.41) SMN1; SMN2RAB9AKMT2ANPC1ALDH1A1
SCHEMBL10701527 0.81 MAPT (0.49) SMN1; SMN2KMT2ANPC1ALDH1A1MEN1
SCHEMBL10699942 0.81 MAPT (0.51) SMN1; SMN2RAB9AKMT2ANPC1MEN1
SCHEMBL10696534 0.81 MAPT (0.42) SMN1; SMN2RAB9AKMT2ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed