SCHEMBL10697104

SCHEMBL10697104

CCCCn1c(=O)c2c(ncn2CC(C)=O)n(Cc2ccccc2)c1=O

nearest known ligand 0.79

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.79
PDE4B Q07343 3/20 0.79
PDE4C Q08493 3/20 0.79
PDE4D Q08499 3/20 0.79
ADORA2A P29274 1/20 0.79
ADORA2B P29275 1/20 0.79
KMT2A Q03164 5/20 0.61
ALDH1A1 P00352 1/20 0.61
CNOT7 Q9UIV1 4/20 0.58
SMN1; SMN2 Q16637 1/20 0.57
MEN1 O00255 3/20 0.57
HPGD P15428 1/20 0.56
TSHR P16473 1/20 0.56
MAPK1 P28482 1/20 0.56
PKM P14618 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10693479 0.89 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL127152 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL7299526 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10695208 0.89 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL11044404 0.88 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10872056 0.87 PDE4A (0.95) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL1946890 0.87 POLB (0.67) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3615415 0.86 ALDH1A1 (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7323464 0.86 PDE4A (0.93) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10694108 0.85 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP disclosed