SCHEMBL10697321

SCHEMBL10697321

COc1c(-c2nc3cc4c(cc3[nH]2)C(C)(C)CNC4=O)ccc(C)c1S

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 9/20 0.45
AURKA O14965 2/20 0.35
KDR P35968 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
ERAP1 Q9NZ08 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MAPKAPK2 P49137 1/20 0.33
NPBWR1 P48145 2/20 0.32
CDC7 O00311 1/20 0.32
AURKB Q96GD4 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705366 0.82 TP53 (0.42) AMY1AAURKAKDRPDE4APDE4B
SCHEMBL10700489 0.79 NPC1 (0.49) AURKAKDRNPC1RAB9APDE4A
SCHEMBL9703298 0.78 PDE5A (0.38) AMY1AAURKAKDRNPC1RAB9A
SCHEMBL9703362 0.77 PDE5A (0.37) AMY1AAURKAKDRPDE4APDE4B
SCHEMBL9383861 0.77 CDK4 (0.41) AMY1APDE3BPDE3ANPBWR1
SCHEMBL10373866 0.77 PDE4A (0.50) AMY1AAURKANPC1RAB9AATM
SCHEMBL10697003 0.77 AMY1A (0.45) AMY1AAURKAKDRNPC1RAB9A
SCHEMBL9703307 0.77 PDE4A (0.34) AMY1AAURKAKDRNPC1RAB9A
SCHEMBL9385702 0.76 PDE4A (0.59) NPC1RAB9APDE4APDE4BPDE4C
SCHEMBL9704386 0.76 PDE2A (0.39) AMY1AAURKAKDRPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0275888-A2 Tricyclic benzimidazoles, process for their preparation and use as medicaments Roche Diagnostics GmbH (DE) 1988-07-27 EP disclosed