SCHEMBL10697003

SCHEMBL10697003

COc1c(-c2nc3cc4c(cc3[nH]2)CC(C)(C)C(=O)N4)ccc(C)c1S

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 9/20 0.45
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
AURKA O14965 2/20 0.36
AURKB Q96GD4 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
ERAP1 Q9NZ08 1/20 0.34
KDR P35968 1/20 0.33
NPBWR1 P48145 3/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 2/20 0.31
POLB P06746 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703536 0.82 TP53 (0.42) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL10373866 0.81 PDE4A (0.50) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL9703372 0.78 AMY1A (0.38) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL9703397 0.77 NPC1 (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9703453 0.77 AMY1A (0.37) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL10697321 0.77 AMY1A (0.45) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL9703459 0.76 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9703379 0.75 PDE4A (0.37) AMY1APDE4APDE4BPDE4CPDE4D
SCHEMBL9378683 0.73 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10700314 0.71 AMY1A (0.48) AMY1APDE3BPDE3ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0275888-A2 Tricyclic benzimidazoles, process for their preparation and use as medicaments Roche Diagnostics GmbH (DE) 1988-07-27 EP disclosed