SCHEMBL10698922

SCHEMBL10698922

COc1ccc(-c2nc3cc4c(cc3n2C)N(CCO)C(=O)C4)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
ALDH1A1 P00352 4/20 0.41
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40
PARP1 P09874 1/20 0.39
CNR2 P34972 1/20 0.38
LMNA P02545 2/20 0.38
CHEK2 O96017 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 2/20 0.37
TSHR P16473 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698291 0.96 HDAC1 (0.42) HDAC1HDAC8ALDH1A1BMPR1BBMPR1A
SCHEMBL10700479 0.90 ALDH1A1 (0.46) ALDH1A1BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL10699753 0.85 KDM4E (0.41) ALDH1A1BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL10701774 0.85 TRIM24 (0.43) ALDH1A1PARP1CNR2LMNACHEK2
SCHEMBL10702791 0.84 BMPR1B (0.42) HDAC1HDAC8BMPR1BBMPR1ATGFBR1
SCHEMBL10700170 0.79 BMPR1B (0.38) HDAC1HDAC8ALDH1A1BMPR1BBMPR1A
SCHEMBL10697520 0.79 HDAC1 (0.42) HDAC1HDAC8ALDH1A1PARP1CNR2
SCHEMBL10700889 0.78 BMPR1B (0.43) HDAC1HDAC8ALDH1A1BMPR1BBMPR1A
SCHEMBL10700455 0.77 HDAC1 (0.42) HDAC1HDAC8ALDH1A1PARP1CNR2
SCHEMBL10698954 0.77 CYP11B1 (0.48) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed