SCHEMBL10705461

SCHEMBL10705461

O=c1ncc2c3c(ccc2[nH]1)OCO3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.42
PDE10A Q9Y233 1/20 0.36
CYP19A1 P11511 2/20 0.35
ACHE P22303 2/20 0.34
CYP1A2 P05177 3/20 0.33
CYP1B1 Q16678 2/20 0.33
TXNRD1 Q16881 1/20 0.33
TXNRD3 Q86VQ6 1/20 0.33
TXNRD2 Q9NNW7 1/20 0.33
CYP1A1 P04798 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
MAPK1 P28482 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
RGS17 Q9UGC6 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10704493 0.70 CA2 (0.49) PDE10AKDM4EMEN1HPGDKMT2A
SCHEMBL19776164 0.69 NQO2 (0.49) NQO2CYP19A1ACHECYP1A2KDM4E
SCHEMBL24149616 0.68 KDM4E (0.48) NQO2CYP1A2KDM4EMEN1ALDH1A1
SCHEMBL32669418 0.67 TTBK1 (0.40) NQO2CYP19A1ACHECYP1A2TXNRD1
SCHEMBL31184823 0.66 ALDH1A1 (0.39) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL3525845 0.65 MAP2K4 (0.45) PDE10AKDM4EMEN1ALDH1A1HPGD
SCHEMBL7215930 0.65 MEN1 (0.35) KDM4EMEN1ALDH1A1LMNAMAPT
SCHEMBL29162197 0.65 DAO (0.39) ACHEKDM4EMEN1ALDH1A1HPGD
SCHEMBL9739366 0.65 NQO2 (0.37) NQO2CYP19A1ACHECYP1A2CYP1B1
SCHEMBL10915643 0.65 NQO2 (0.41) NQO2PDE10ACYP19A1TXNRD1TXNRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0138490-B1 4-alkyl methylenedioxy-2-1[H]-quinazolinones ORTHO PHARMACEUTICAL CORPORATION (US) 1988-04-27 EP disclosed
US-4617392-A 4-alkyl-5,6-methylenedioxy-2-1[H]-quinazolinones useful as cardiotonic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1986-10-14 US disclosed
EP-0138490-A1 4-alkyl methylenedioxy-2-1[H]-quinazolinones ORTHO PHARMACEUTICAL CORPORATION (US) 1985-04-24 EP disclosed