SCHEMBL10707249

SCHEMBL10707249

CC(C)(C)OC(=O)N(CC(=O)OCc1ccccc1)C(=O)[C@@H](N)Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.46
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
CTSL P07711 3/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 3/20 0.41
NR1D1 P20393 1/20 0.40
MMP2 P08253 1/20 0.40
SLC15A1 P46059 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPC1 O15118 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ANPEP P15144 1/20 0.39
ERAP2 Q6P179 1/20 0.39
ERAP1 Q9NZ08 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11210582 0.88 MC4R (0.51) MC4RITGA4ITGB7CTSLALDH1A1
SCHEMBL13150768 0.78 L3MBTL1 (0.43) ITGA4ITGB7ALDH1A1SLC15A1
SCHEMBL29077734 0.77 L3MBTL1 (0.50) ALDH1A1MAPTKMT2ATDP1
SCHEMBL5724173 0.77 ALDH1A1 (0.54) ALDH1A1MAPTRAB9ANR1D1
SCHEMBL7737719 0.76 RAB9A (0.55) MC4RITGA4ITGB7CTSLRAB9A
SCHEMBL5724430 0.76 ALDH1A1 (0.48) ALDH1A1MAPTRAB9ANR1D1MMP2
SCHEMBL9706834 0.75 MC4R (0.51) MC4RITGA4ITGB7CTSLRAB9A
SCHEMBL8251477 0.75 ITGA4 (0.49) MC4RITGA4ITGB7ALDH1A1MAPT
SCHEMBL2502338 0.75 ITGA4 (0.49) MC4RITGA4ITGB7ALDH1A1MAPT
SCHEMBL10598042 0.73 HTR2A (0.41) MC4RITGA4ITGB7CTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0117089-B1 BETA-ADRENERGIC ANTAGONIST COMPOUNDS AND DERIVATIVES OF BETA-ADRENERGIC ANTAGONISTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1988-12-14 EP disclosed