SCHEMBL1072250

SCHEMBL1072250

C[C@@](N=C=O)(C(=O)O)C1CCCCC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
EPHX1 P07099 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
SSTR4 P31391 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1260690 0.98 KEAP1 (0.33) ALDH1A1EPHX1KEAP1NFE2L2
SCHEMBL29889579 0.75 KEAP1 (0.35) EPHX1KEAP1NFE2L2SSTR4
SCHEMBL4310017 0.74 ALDH1A1 (0.39) ALDH1A1SSTR4
SCHEMBL9795387 0.74 ALDH1A1 (0.39) ALDH1A1
SCHEMBL8196191 0.74 KEAP1 (0.33) ALDH1A1KEAP1NFE2L2
SCHEMBL4209005 0.71 ALDH1A1 (0.37) ALDH1A1
SCHEMBL10790172 0.71 ALDH1A1 (0.37) ALDH1A1
SCHEMBL1876976 0.69 EPHX1 (0.39) ALDH1A1EPHX1KEAP1NFE2L2SSTR4
SCHEMBL29122810 0.69 EPHX1 (0.39) ALDH1A1EPHX1KEAP1NFE2L2SSTR4
SCHEMBL2895430 0.69 ALDH1A1 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110002884-A1 THERAPEUTIC COMPOUNDS MERCK SHARP & DOHME LLC 2011-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110002884-A1 THERAPEUTIC COMPOUNDS RRP1B, ZC3HAV1, RNASE1 ALDH1A1 1039/4885EPHX1 1536/4885KEAP1 290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.