SCHEMBL10732292

SCHEMBL10732292

Cc1ncc2c(c1O)COC2C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
P2RX3 P56373 1/20 0.42
KMT2A Q03164 1/20 0.42
ADRA2A P08913 4/20 0.33
ADRA2B P18089 4/20 0.33
ADRA2C P18825 4/20 0.33
ADRA1D P25100 4/20 0.33
ADRA1A P35348 4/20 0.33
ADRA1B P35368 4/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10830005 0.79 ADRA2A (0.39) KDM4EMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL10737643 0.79 ADRA2A (0.33) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9751410 0.79 KDM4E (0.39) KDM4EMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL11563119 0.78 KDM4E (0.41) KDM4EMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL10821406 0.78 PDXK (0.38) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10734345 0.78 ADRA2A (0.33) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10830702 0.76 CYP2D6 (0.38) KDM4EMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL10842038 0.76 ADRA2A (0.40) KDM4EMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL10820964 0.75 ADRA2A (0.40) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11134644 0.75 SLC5A2 (0.39) KDM4EMEN1CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4659719-A CALCIUM OR SEROTONIN ANTAGONIST SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1987-04-21 US disclosed
US-4585776-A DIURETIC HYPOTENSIVE SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1986-04-29 US disclosed
US-4383998-A Furo-(3,4-c)-pyridine derivatives and their pharmaceutical use SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (FR) 1983-05-17 US disclosed