SCHEMBL10749867

SCHEMBL10749867

c1ccc2[nH]c(NC3CCN(CCNn4nccn4)CC3)nc2c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.59
TSHR P16473 2/20 0.50
BACE1 P56817 1/20 0.42
CHRNA7 P36544 1/20 0.42
HDAC6 Q9UBN7 1/20 0.40
KCNN3 Q9UGI6 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
JAK1 P23458 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1151915 0.83 KCNH2 (0.59) KCNH2TSHRBACE1CHRNA7HDAC6
SCHEMBL9698375 0.82 KCNH2 (0.66) KCNH2TSHRCHRNA7HDAC6KCNN3
SCHEMBL11266594 0.80 KCNH2 (0.80) KCNH2TSHRCHRNA7GAAJAK1
SCHEMBL7416758 0.79 KCNH2 (0.65) KCNH2TSHRHDAC6KCNN3JAK1
SCHEMBL10508648 0.79 KCNH2 (0.55) KCNH2TSHRBACE1CHRNA7KDM4E
SCHEMBL8562586 0.78 KCNH2 (0.65) KCNH2TSHRCHRNA7
Water SCHEMBL8562628 0.77 KCNH2 (0.61) KCNH2HDAC6KCNN3
Water SCHEMBL8566156 0.77 KCNH2 (0.61) KCNH2HDAC6KCNN3
SCHEMBL8560605 0.77 KCNH2 (0.61) KCNH2HDAC6KCNN3
SCHEMBL3748349 0.77 KCNH2 (0.63) KCNH2BACE1KDM4EGAAJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4634704-A HISTAMINE AND SEROTONINE ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 1987-01-06 US disclosed