SCHEMBL10758591

SCHEMBL10758591

O=C(O)CC(=O)CCCc1ccccc1OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 7/20 0.60
PTGER4 P35408 7/20 0.60
PTGER3 P43115 7/20 0.60
PTGER2 P43116 7/20 0.60
HTR1A P08908 1/20 0.56
DRD2 P14416 1/20 0.56
MGLL Q99685 1/20 0.53
FOLH1 Q04609 1/20 0.51
ABCB1 P08183 2/20 0.49
GAA P10253 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
HPGD P15428 1/20 0.47
BLM P54132 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990040 0.83 PTGER1 (0.60) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL2038509 0.82 PTGER1 (0.67) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL17197391 0.80 HTR1A (0.79) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL8676328 0.80 PTGER1 (0.59) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL10753679 0.79 FFAR1 (0.68) TDP1
SCHEMBL7425846 0.77 MEN1 (0.60) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL31561714 0.77 HTR1A (0.69) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL3159332 0.77 HTR1A (0.69) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL3930253 0.77 HTR1A (0.59) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL8675205 0.77 PTGER1 (0.71) PTGER1PTGER4PTGER3PTGER2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4672071-A Antihypertensive dihydropyridine compositions, optical isomers and intermediates SYNTEX (U.S.A.) INC. (US) 1987-06-09 US disclosed
EP-0191448-A2 Antihypertensive dihydropyridine derivatives SYNTEX (U.S.A.) INC. (US) 1986-08-20 EP disclosed
US-4595690-A Hypotensive agents SYNTEX (U.S.A.) INC. (US) 1986-06-17 US disclosed